Procaine-CAS 59-46-1
Procaine / Procaine Hydrochloride yog dab tsi?
Procaine HCl yog ib qho tshuaj loog hauv zos ntawm cov amino ester pawg. Nws yog siv ua ntej kom txo tau qhov mob ntawm kev txhaj tshuaj ntawm penicillin, thiab nws kuj yog siv hauv kev kho hniav. Nws feem ntau ua los ntawm kev ua sodium sodium blocker. Niaj hnub no nws tau siv kho nyob rau hauv qee lub teb chaws vim nws cov sympatholytic, tiv thaiv kev mob, kev ua kom zoo dua, thiab mus ob peb vas kho qhov teebmeem.
Procaine HCl yog qhia rau kev tsim cov tshuaj loog hauv zos lossis ib cheeb tsam thiab kev ua kom loog los ntawm kev nkag rau hauv zos thiab peripheral hlab ntaws cov tswv yim.
Khoom Npe | Khoom Siv Procaine / Procaine Hydrochloride |
Cas | 51-05-8 / 59-46-1 |
Tsos | dawb crystalline hmoov |
Molecular Luj | 272.77 |
Ntsuas | 98% |
Txee Lub Neej | 24 lub hlis thaum cia zoo |
Cia | Khaws rau hauv qhov chaw txias, qhuav, thiab tsaus |
Thov
Procaine HCl yog ib qho tshuaj loog hauv zos ntawm cov amino ester pawg. Nws yog siv ua ntej kom txo tau qhov mob ntawm kev txhaj tshuaj ntawm penicillin, thiab nws kuj yog siv hauv kev kho hniav. Los ntawm qhov ubiquity ntawm lub lag luam npe Novocain, nyob rau qee thaj tsam procaine raug xa mus rau generically Nws ua feem ntau yog los ntawm sodium sodium blocker.Today nws siv kho nyob rau qee lub tebchaws vim nws cov sympatholytic, anti-inflammatory, perfusion txhim kho, thiab mus ob peb vas txhim kho cov teebmeem.
Procaine HCl yog qhia rau kev tsim cov tshuaj loog hauv zos lossis ib cheeb tsam thiab kev ua kom loog los ntawm kev nkag rau hauv zos thiab peripheral hlab ntaws cov tswv yim.
Daim ntawv thov ntawm procaine ua rau kev nyuaj siab ntawm kev ua tsis tau neuronal. Qhov kev ntxhov siab ua rau cov hlab hlwb ua rau lub ntsej muag tsis txaus siab thiab ua kom lub cev tsis haum thiab ua rau lub siab mos, ua rau muaj hnub nyoog mus rau qhov pom tseeb ceev. Cov kev tshawb fawb txog tsiaj tau qhia txog kev siv cov procaine ua rau muaj kev nce ntawm dopamine thiab serotonin ntau ntau hauv lub hlwb.Lub teeb meem ntau ntxiv yuav tshwm sim vim kev sib txawv ntawm tib neeg ua siab ntev rau procaine
tsuas tshuaj. Kev poob siab thiab kiv taub hau tuaj yeem tshwm sim los ntawm qhov kev zam ntawm lub hauv nruab nrab lub paj hlwb, uas tuaj yeem ua rau ua pa tsis ua haujlwm yog tias dhau sijhawm. Procaine kuj tseem tseem ua rau lub zog myocardium ua rau lub plawv dhia tsis zoo.
Procaine tseem tuaj yeem ua rau muaj kev tsis haum tshuaj ua rau cov tib neeg muaj teeb meem ua pa, tawm pob, thiab o. Cov kev tsis haum rau procaine feem ntau tsis yog teb rau procaine nws tus kheej, tab sis rau nws qhov metabolite PABA. Muaj li ntawm ib ntawm 3000 tus neeg muaj ib daim ntawv atypical pseudocholinesterase, [citation ntxiv] uas tsis hydrolyze ester cov tshuaj loog xws li procaine, uas ua rau lub sijhawm ntev
ntawm theem siab ntawm cov tshuaj loog hauv cov ntshav thiab muaj cov tshuaj lom ntau ntxiv.